BChE

BChE產(chǎn)品

所有產(chǎn)品(7)
BChE抑制劑 (7)
新BChE產(chǎn)品

目錄號(hào)	產(chǎn)品名	產(chǎn)品描述
S0924	Pteryxin	Pteryxin ((+)-Pteryxin) 是一種在 Apiaceae 傘形科中發(fā)現(xiàn)的二氫吡喃香豆素衍生物，也是一種有效的 butyrylcholinesterase (BChE) 的抑制劑，IC50值為12.96 μg/ml。Pteryxin 可抑制LPS誘導(dǎo)的小鼠腹膜巨噬細(xì)胞中 nitric oxide 的產(chǎn)生，其IC50值為20 μM。Pteryxin 具有治療阿爾茨海默氏病 (AD) 的潛力。
S3245	Nodakenetin	Nodakenetin (NANI) 是從Angelica decursiva中分離出的植物性香豆素，可抑制 α-glucosidase、PTP1B、rat lens aldose reductase (RLAR)、AChE、BChE 和 β-site amyloid precursor protein cleaving enzyme 1 (BACE1)。Nodakenetin 可改變 Bax 和 Bcl-2 的蛋白質(zhì)表達(dá)，并促進(jìn)線粒體凋亡。Nodakenetin 具有抗腫瘤活性。
S5665	Drofenine Hydrochloride	Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers.
S3835	Loganin	Loganin (Loganoside) is an iridoid glycoside first isolated from the seeds of Strychnos nux-vomica, a member of the Loganiaceae family. It is a non-competitive inhibitor of BACE1 with IC50 of 47.97 μM an also inhibits AChE and BChE with IC50 values of 3.95 μM and 33.02 μM, respectively.
E2237	Vasicine (hydrochloride)	Vasicine hydrochloride(Peganine hydrochloride)是一種從Adhatoda vasica中分離出來的生物堿vasicine (VAS)的鹽，是一種潛在的天然膽堿酯酶抑制劑。VAS抑制乙酰膽堿酯酶(AChE)和丁酰膽堿酯酶(BChE)。
S5511	Ethyl (triphenylphosphoranylidene) acetate	Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
E0784	MAO-B-IN-2	MAO-B-in-2是MAO-B和BChE的選擇性，競(jìng)爭(zhēng)性抑制劑，其IC50分別為0.51和7.00 μM。
S0924	Pteryxin	Pteryxin ((+)-Pteryxin) 是一種在 Apiaceae 傘形科中發(fā)現(xiàn)的二氫吡喃香豆素衍生物，也是一種有效的 butyrylcholinesterase (BChE) 的抑制劑，IC50值為12.96 μg/ml。Pteryxin 可抑制LPS誘導(dǎo)的小鼠腹膜巨噬細(xì)胞中 nitric oxide 的產(chǎn)生，其IC50值為20 μM。Pteryxin 具有治療阿爾茨海默氏病 (AD) 的潛力。
S3245	Nodakenetin	Nodakenetin (NANI) 是從Angelica decursiva中分離出的植物性香豆素，可抑制 α-glucosidase、PTP1B、rat lens aldose reductase (RLAR)、AChE、BChE 和 β-site amyloid precursor protein cleaving enzyme 1 (BACE1)。Nodakenetin 可改變 Bax 和 Bcl-2 的蛋白質(zhì)表達(dá)，并促進(jìn)線粒體凋亡。Nodakenetin 具有抗腫瘤活性。
S5665	Drofenine Hydrochloride	Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers.
S3835	Loganin	Loganin (Loganoside) is an iridoid glycoside first isolated from the seeds of Strychnos nux-vomica, a member of the Loganiaceae family. It is a non-competitive inhibitor of BACE1 with IC50 of 47.97 μM an also inhibits AChE and BChE with IC50 values of 3.95 μM and 33.02 μM, respectively.
E2237	Vasicine (hydrochloride)	Vasicine hydrochloride(Peganine hydrochloride)是一種從Adhatoda vasica中分離出來的生物堿vasicine (VAS)的鹽，是一種潛在的天然膽堿酯酶抑制劑。VAS抑制乙酰膽堿酯酶(AChE)和丁酰膽堿酯酶(BChE)。
S5511	Ethyl (triphenylphosphoranylidene) acetate	Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
E0784	MAO-B-IN-2	MAO-B-in-2是MAO-B和BChE的選擇性，競(jìng)爭(zhēng)性抑制劑，其IC50分別為0.51和7.00 μM。