| S9668 |
PKR-IN-C16
|
PKR-IN-C16 (C16, Imidazolo-oxindole PKR inhibitor C16) 是一種RNA-dependent protein kinase (PKR, Protein Kinase R, EIF2AK2)的特異性抑制劑。PKR-IN-C16 可在具有神經(jīng)炎癥成分的急性興奮性毒性大鼠模型中阻止凋亡和 IL-1β 的產(chǎn)生。 |
-
Immunity, 2025, 58(10):2489-2504.e8
-
Exp Mol Med, 2024, 56(2):408-421.
-
EMBO J, 2024, 43(5):780-805.
|
|
| S6508 |
Mitapivat
|
Mitapivat (AG-348)是丙酮酸激酶PKM2的激活劑。PKM2參與糖酵解。 |
-
Proc Natl Acad Sci U S A, 2022, 119(40):e2210779119
|
|
| F1207 |
PKR Antibody [K23G2]
|
|
|
|
| F1597 |
Phospho-PKR (Thr446) Antibody [K16N13]
|
|
|
|
| F2996New |
PACT (PKR activating protein) / PRKRA Antibody [F4M5]
|
PACT,PACT (PKR activating protein) / PRKRA |
|
|
| E2388 |
PKR-IN-2
|
PKR-IN-2是從專利WO2014139144A1中提取的丙酮酸激酶同種型PKR激活劑,化合物160;PKR- IN -2可用于PKR功能相關(guān)疾病的研究,包括癌癥、糖尿病、肥胖、自身免疫性疾病、良性前列腺增生等。 |
|
|