| S0141 |
NQ301
|
NQ301 (Compound 211) 是一種抗血小板和抗血栓形成劑,也是一種選擇性的 CD45 的抑制劑,IC50值為200 nM。NQ301 可抑制兔血小板中的 thromboxane A2 receptor (TXA2) 和合酶synthase的活性。 |
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J Extracell Vesicles, 2021, 10(5):e12078
|
|
| S4495 |
Quinine
|
Quinine 是一種來自cinchona tree的生物堿,是一種抗瘧疾劑和鉀通道 potassium channel 的抑制劑,可抑制電壓誘發(fā)的mSlo3 (KCa 5.1)通道電流,脈沖至+100 mV,其IC50值為169 μM。[2] |
-
Cell Mol Immunol, 2022, 19(8):925-943
-
J Pharmacol Toxicol Methods, 2017, 90:39-47
|
|
| S5271 |
Suloctidil
|
Suloctidil, a sulfur-containing aminoalcohol showing to inhibit human platelet aggregation, is a peripheral vasodilator and a potential antifungal agent. |
|
|
| S9360 |
4-Hydroxyquinazoline
|
4-Hydroxyquinazoline (Quinazolin-4-ol, 4-Quinazolinol) 是 PARP 的抑制劑,對 PARP-1 的IC50值為9.5 μM。 |
|
|
| S3711 |
Carbasalate Calcium
|
Carbasalate calcium (Iromin, Alcacyl, Omegin, Rheomin, Solupsan) 是一種止痛劑、退熱劑,是一種抗炎藥物以及血小板聚集的抑制劑。 |
|
|
| S3883 |
Protopine
|
Protopine (Corydinine, Fumarine, Biflorine, Macleyine), an alkaloid present in different plants, has been shown to exhibit a number of activities, such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation. It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities. |
|
|
| S4492 |
Dextran
|
Dextran (Dextran 40, Macrodex) 是一種具有生物相容性、無毒且無免疫原性的生物物質,已廣泛用于給藥體系。 |
|
|
| S0141 |
NQ301
|
NQ301 (Compound 211) 是一種抗血小板和抗血栓形成劑,也是一種選擇性的 CD45 的抑制劑,IC50值為200 nM。NQ301 可抑制兔血小板中的 thromboxane A2 receptor (TXA2) 和合酶synthase的活性。 |
- J Extracell Vesicles, 2021, 10(5):e12078
|
|
| S4495 |
Quinine
|
Quinine 是一種來自cinchona tree的生物堿,是一種抗瘧疾劑和鉀通道 potassium channel 的抑制劑,可抑制電壓誘發(fā)的mSlo3 (KCa 5.1)通道電流,脈沖至+100 mV,其IC50值為169 μM。[2] |
- Cell Mol Immunol, 2022, 19(8):925-943
- J Pharmacol Toxicol Methods, 2017, 90:39-47
|
|
| S5271 |
Suloctidil
|
Suloctidil, a sulfur-containing aminoalcohol showing to inhibit human platelet aggregation, is a peripheral vasodilator and a potential antifungal agent. |
|
|
| S9360 |
4-Hydroxyquinazoline
|
4-Hydroxyquinazoline (Quinazolin-4-ol, 4-Quinazolinol) 是 PARP 的抑制劑,對 PARP-1 的IC50值為9.5 μM。 |
|
|
| S3711 |
Carbasalate Calcium
|
Carbasalate calcium (Iromin, Alcacyl, Omegin, Rheomin, Solupsan) 是一種止痛劑、退熱劑,是一種抗炎藥物以及血小板聚集的抑制劑。 |
|
|
| S3883 |
Protopine
|
Protopine (Corydinine, Fumarine, Biflorine, Macleyine), an alkaloid present in different plants, has been shown to exhibit a number of activities, such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation. It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities. |
|
|