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    • Platelet aggregation

      Platelet aggregation產(chǎn)品

      • 所有產(chǎn)品(7)
      • Platelet aggregation抑制劑 (6)
      目錄號 產(chǎn)品名 產(chǎn)品描述 文獻引用 實驗數(shù)據(jù)
      S0141 NQ301 NQ301 (Compound 211) 是一種抗血小板和抗血栓形成劑,也是一種選擇性的 CD45 的抑制劑,IC50值為200 nM。NQ301 可抑制兔血小板中的 thromboxane A2 receptor (TXA2) 和合酶synthase的活性。
      J Extracell Vesicles, 2021, 10(5):e12078
      S4495 Quinine Quinine 是一種來自cinchona tree的生物堿,是一種抗瘧疾劑和鉀通道 potassium channel 的抑制劑,可抑制電壓誘發(fā)的mSlo3 (KCa 5.1)通道電流,脈沖至+100 mV,其IC50值為169 μM。[2]

      Cell Mol Immunol, 2022, 19(8):925-943
      J Pharmacol Toxicol Methods, 2017, 90:39-47
      S5271 Suloctidil Suloctidil, a sulfur-containing aminoalcohol showing to inhibit human platelet aggregation, is a peripheral vasodilator and a potential antifungal agent.
      S9360 4-Hydroxyquinazoline 4-Hydroxyquinazoline (Quinazolin-4-ol, 4-Quinazolinol) 是 PARP 的抑制劑,對 PARP-1 的IC50值為9.5 μM。
      S3711 Carbasalate Calcium Carbasalate calcium (Iromin, Alcacyl, Omegin, Rheomin, Solupsan) 是一種止痛劑、退熱劑,是一種抗炎藥物以及血小板聚集的抑制劑。
      S3883 Protopine Protopine (Corydinine, Fumarine, Biflorine, Macleyine), an alkaloid present in different plants, has been shown to exhibit a number of activities, such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation. It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities.
      S4492 Dextran Dextran (Dextran 40, Macrodex) 是一種具有生物相容性、無毒且無免疫原性的生物物質,已廣泛用于給藥體系。
      S0141 NQ301 NQ301 (Compound 211) 是一種抗血小板和抗血栓形成劑,也是一種選擇性的 CD45 的抑制劑,IC50值為200 nM。NQ301 可抑制兔血小板中的 thromboxane A2 receptor (TXA2) 和合酶synthase的活性。
      J Extracell Vesicles, 2021, 10(5):e12078
      S4495 Quinine Quinine 是一種來自cinchona tree的生物堿,是一種抗瘧疾劑和鉀通道 potassium channel 的抑制劑,可抑制電壓誘發(fā)的mSlo3 (KCa 5.1)通道電流,脈沖至+100 mV,其IC50值為169 μM。[2]

      Cell Mol Immunol, 2022, 19(8):925-943
      J Pharmacol Toxicol Methods, 2017, 90:39-47
      S5271 Suloctidil Suloctidil, a sulfur-containing aminoalcohol showing to inhibit human platelet aggregation, is a peripheral vasodilator and a potential antifungal agent.
      S9360 4-Hydroxyquinazoline 4-Hydroxyquinazoline (Quinazolin-4-ol, 4-Quinazolinol) 是 PARP 的抑制劑,對 PARP-1 的IC50值為9.5 μM。
      S3711 Carbasalate Calcium Carbasalate calcium (Iromin, Alcacyl, Omegin, Rheomin, Solupsan) 是一種止痛劑、退熱劑,是一種抗炎藥物以及血小板聚集的抑制劑。
      S3883 Protopine Protopine (Corydinine, Fumarine, Biflorine, Macleyine), an alkaloid present in different plants, has been shown to exhibit a number of activities, such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation. It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities.
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