• <dfn id="q240u"></dfn>
      • CDK1
      • CDK2
      • CDK3
      • CDK4
      • CDK5
      • CDK6
      • CDK7
      • CDK9
      • CLK
      • Cdc
      • CDK8
      • CDK12
      • CDK13
      • CDK19
      • CDK11
      • CDK/cyclin complexes

      CLK 選擇性抑制劑

      目錄號(hào) 產(chǎn)品名 產(chǎn)品描述 Selective / Pan IC50 / Ki
      S6768 CC-671 CC-671 is a selectively dual inhibitor of TTK (human protein kinase monopolar spindle 1 [hMps1]) and CDC like kinase 2 (CLK2) with IC50s of 5 nM and 3 nM for TTK and CLK2, respectively. Selective CLK2, IC50: 3 nM
      S7320 TG003 TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC. Selective mCLK1, IC50: 20 nM; mCLK2, IC50: 200 nM; mCLK4, IC50: 15 nM
      S7509 ML167 ML167 (CID 44968231) is a highly selective Cdc2-like kinase 4 (Clk4) inhibitor with IC50 of 136 nM, >10-fold selectivity for closely related kinases Clk1-3 and Dyrk1A/1B. Selective CLK4, IC50: 136 nM; CLK1, IC50: 1522 nM; CLK2, IC50: 1648 nM; Dyrk1B , IC50: 4420 nM
      在線咨詢(xún)
      聯(lián)系我們
        • <dfn id="q240u"></dfn>
        • 性生活免费片 | 中文字幕av在线观看 | www.蜜乳av.com | 欧美精品性 | 日本久久不卡视频 |