PDE4B 抑制劑
| 目錄號 |
產品名 |
產品描述 |
Selective / Pan |
IC50 / Ki |
| S2620 |
GSK256066 |
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2. |
Pan |
PDE4B, IC50: 3.2 pM |
| S1430 |
Rolipram (ZK-62711) |
The PDE4 selective inhibitor, Rolipram (ZK-62711, SB 95952), inhibited immunopurified PDE4B and PDE4D activities similarly, with IC50 values of approx. 130 nM and 240 nM respectively; an anti-inflammatory agent. |
Pan |
PDE4B, IC50: 130 nM |
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