| S7497 |
CK-636
|
CK-636 (CK-0944636)是一種Arp2/3復(fù)合抑制劑,其IC50為4 μM,在24 μM 和 32 μM時(shí),分別能夠抑制人的肌動(dòng)蛋白聚合誘導(dǎo)和裂殖酵母與bovine Arp2/3的復(fù)合物。 |
-
J Biol Chem, 2024, 300(12):107942
-
Elife, 2021, 10e65910
-
Theranostics, 2019, 9(25):7628-7647
|
|
| S8184 |
Cytochalasin D
|
Cytochalasin D (Zygosporin A, NSC 209835) 是一種源自真菌的有效肌動(dòng)蛋白聚合抑制劑。 Cytochalasin D抑制細(xì)胞中肌動(dòng)蛋白絲的動(dòng)力學(xué)。 它誘導(dǎo) Yap 磷酸化和細(xì)胞質(zhì)滯留。 |
-
Nat Commun, 2025, 16(1):4069
-
Cell Regen, 2025, 14(1):21
-
Cell Prolif, 2024, e13728.
|
|
| S5256 |
Benproperine phosphate
|
Benproperine phosphate (Blascorid, Pirexyl) 是一種止咳藥,一種口服活性的 actin-related protein 2/3 complex subunit 2 (ARPC2) 的有效抑制劑。Benproperine phosphate 會(huì)削弱 Arp2/3 功能,從而減弱肌動(dòng)蛋白actin的聚合成核速率。Benproperine phosphate 可抑制癌細(xì)胞遷移和腫瘤轉(zhuǎn)移。 |
-
Mol Oncol, 2020, 10.1002/1878-0261.12854
|
|
| F0012 |
β-Actin Antibody [C21N23]
|
ACTB,beta Actin,beta Actin Loading Control,beta-Actin,β-Actin |
-
Adv Sci (Weinh), 2025, 12(35):e05725
-
Cell Death Dis, 2025, 16(1):672
-
J Agric Food Chem, 2025, 73(50):31893-31905
|
|
| F0017 |
α-Smooth Muscle Actin Antibody [L19D14]
|
Actin, alpha-Smooth Muscle,Actin, α-Smooth Muscle,alpha smooth muscle Actin,Alpha-Smooth Muscle Actin,Smooth Muscle Actin,α-Actin,α-Smooth Muscle Actin, α-SMA, a-SMA |
-
Bioact Mater, 2024, 34:51-63
-
J Plast Surg Hand Surg, 2021, 55(5):284-293
|
|
| F0082 |
Actin Antibody [A24J5]
|
Actin Rabbit mAb recognizes endogenous levels of total Actin protein. |
|
|
| F0440 |
Neurofilament-L Antibody [L10B15]
|
68kDa Neurofilament/NF-L,Neurofilament 68,Neurofilament 70 kDa,Neurofilament-L,NF-L |
|
|
| F0695 |
Neurofilament-M Antibody [H7L9]
|
160 kD Neurofilament Medium,NEFM,Neurofilament 145 kDa,Neurofilament 160,Neurofilament 160 kDa,Neurofilament M,Neurofilament-M |
|
|
| F1648 |
PABP1 Antibody [H6J19]
|
PABP, PABP1 |
|
|
| F0278 |
Cofilin Antibody [D9A5]
|
Cofilin,Cofilin 1 |
|
|
| F2199 |
α Actinin 1/ACTN1 Antibody [C8H2]
|
Actinin alpha,alpha Actinin/ACTN1,alpha-Actinin,α-Actinin |
|
|
| F2226 |
α smooth muscle Actin (acetyl Glu 3) + Actin γ2 (acetyl Glu3) Antibody [H16P9]
|
|
|
|
| F0640 |
N-WASP Antibody [K15N2]
|
N WASP,N-WASP |
|
|
| F0417 |
VASP Antibody [A20G16]
|
|
|
|
| F1962 |
Phospho-Lamin A/C (Ser22) Antibody [D12F9]
|
|
|
|
| F1379 |
Tropomyosin-1 Antibody [G4H1]
|
Tropomyosin (Sarcomeric),Tropomyosin-1 |
|
|
| F2176 |
SUN2 Antibody [D3P18]
|
|
|
|
| F2446 |
γ Actin Antibody [A4H18]
|
gamma Actin,gamma-Actin |
|
|
| F2365 |
Arp3 C-terminal Antibody [F20N23]
|
|
|
|
| F2091 |
Fascin Antibody [N3C10]
|
|
|
|
| F2612 |
ARPC2 Antibody [B10F4]
|
ARPC2,p34-Arc/ARPC2 |
|
|
| F2033 |
α Actinin 4 Antibody [D15C11]
|
alpha Actinin 4,α-Actinin 4 |
|
|
| F2681 |
Cytokeratin 5 Antibody [G20N20]
|
Cytokeratin 5 |
|
|
| F2188 |
Cytokeratin 13 Antibody [L12L19]
|
|
|
|
| F2756 |
CCT2 Antibody [C14D6]
|
|
|
|
| F1440 |
Gelsolin Antibody [D8P23]
|
|
|
|
| F1636 |
Phospho-RAB10 (Thr73) Antibody [M19N14]
|
|
|
|
| F1478 |
Phospho-Zyxin (Ser142/143) Antibody [L24L6]
|
|
|
|
| E1042 |
SMIFH2
|
SMIFH2 是一種特定的 formin 抑制劑,可在體外抑制 formin 驅(qū)動(dòng)的肌動(dòng)蛋白聚合,對(duì)于不同形式formin的 IC50 范圍為 5 mM 至 15 μM。 |
-
Sci Rep, 2025, 15(1):34331
|
|
| S6673 |
CCG-222740
|
CCG-222740是一種Rho/MRTF通路抑制劑。CCG-222740通過降低α平滑肌肌動(dòng)蛋白(alpha smooth muscle actin, α-SMA)的表達(dá)水平來降低星狀細(xì)胞在體外和體內(nèi)的活化。 |
|
|
| E0076 |
Simufilam dihydrochloride
|
Simufilam (PTI-125) Dihydrochloride 是一種小分子調(diào)節(jié)劑,可優(yōu)先結(jié)合改變的 FLNA 并恢復(fù)其天然構(gòu)象,恢復(fù)受體和突觸活動(dòng),并減少其 α7nAChR/TLR4 關(guān)聯(lián)和下游病理。 |
|
|
| E2956 |
Cytochalasin C
|
Cytochalasin C是一種在 C. globosum 中發(fā)現(xiàn)的細(xì)胞滲透性真菌代謝物,是肌動(dòng)蛋白聚合的抑制劑。 它誘導(dǎo)核小棒的形成。 |
|
|
| S3206 |
5a-Pregnane-3,20-dione
|
5a-Pregnane-3,20-dione (5alphaP, 5-a-dihydroprogesterone, 3,20-allopregnanedione, 5-Alpha-Dihydro Progesterone) 是一種內(nèi)源性的孕酮代謝物。5a-Pregnane-3,20-dione 可使肌動(dòng)蛋白actin解聚,并降低 actin 和 vinculin 的表達(dá)。5a-Pregnane-3,20-dione 可通過影響粘附和細(xì)胞骨架分子來參與促進(jìn)乳腺瘤形成和轉(zhuǎn)移。 |
|
|
| S7690 |
CK-666
|
CK-666 是肌動(dòng)蛋白相關(guān)蛋白 2/3 (actin-related protein 2/3, Arp2/3) 復(fù)合物的抑制劑,對(duì) BtArp2/3 復(fù)合物和 SpArp2/3 復(fù)合物的 IC50 分別為 17 μM 和 5 μM。 |
-
Sci Rep, 2025, 15(1):34331
-
Res Sq, 2023, rs.3.rs-3372987
|
|
| F2616 |
Cytokeratin 4 Antibody [G16J4]
|
|
|
|
| S7497 |
CK-636
|
CK-636 (CK-0944636)是一種Arp2/3復(fù)合抑制劑,其IC50為4 μM,在24 μM 和 32 μM時(shí),分別能夠抑制人的肌動(dòng)蛋白聚合誘導(dǎo)和裂殖酵母與bovine Arp2/3的復(fù)合物。 |
- J Biol Chem, 2024, 300(12):107942
- Elife, 2021, 10e65910
- Theranostics, 2019, 9(25):7628-7647
|
|
| S8184 |
Cytochalasin D
|
Cytochalasin D (Zygosporin A, NSC 209835) 是一種源自真菌的有效肌動(dòng)蛋白聚合抑制劑。 Cytochalasin D抑制細(xì)胞中肌動(dòng)蛋白絲的動(dòng)力學(xué)。 它誘導(dǎo) Yap 磷酸化和細(xì)胞質(zhì)滯留。 |
- Nat Commun, 2025, 16(1):4069
- Cell Regen, 2025, 14(1):21
- Cell Prolif, 2024, e13728.
|
|
| S5256 |
Benproperine phosphate
|
Benproperine phosphate (Blascorid, Pirexyl) 是一種止咳藥,一種口服活性的 actin-related protein 2/3 complex subunit 2 (ARPC2) 的有效抑制劑。Benproperine phosphate 會(huì)削弱 Arp2/3 功能,從而減弱肌動(dòng)蛋白actin的聚合成核速率。Benproperine phosphate 可抑制癌細(xì)胞遷移和腫瘤轉(zhuǎn)移。 |
- Mol Oncol, 2020, 10.1002/1878-0261.12854
|
|
| E1042 |
SMIFH2
|
SMIFH2 是一種特定的 formin 抑制劑,可在體外抑制 formin 驅(qū)動(dòng)的肌動(dòng)蛋白聚合,對(duì)于不同形式formin的 IC50 范圍為 5 mM 至 15 μM。 |
- Sci Rep, 2025, 15(1):34331
|
|
| S6673 |
CCG-222740
|
CCG-222740是一種Rho/MRTF通路抑制劑。CCG-222740通過降低α平滑肌肌動(dòng)蛋白(alpha smooth muscle actin, α-SMA)的表達(dá)水平來降低星狀細(xì)胞在體外和體內(nèi)的活化。 |
|
|
| E2956 |
Cytochalasin C
|
Cytochalasin C是一種在 C. globosum 中發(fā)現(xiàn)的細(xì)胞滲透性真菌代謝物,是肌動(dòng)蛋白聚合的抑制劑。 它誘導(dǎo)核小棒的形成。 |
|
|
| S3206 |
5a-Pregnane-3,20-dione
|
5a-Pregnane-3,20-dione (5alphaP, 5-a-dihydroprogesterone, 3,20-allopregnanedione, 5-Alpha-Dihydro Progesterone) 是一種內(nèi)源性的孕酮代謝物。5a-Pregnane-3,20-dione 可使肌動(dòng)蛋白actin解聚,并降低 actin 和 vinculin 的表達(dá)。5a-Pregnane-3,20-dione 可通過影響粘附和細(xì)胞骨架分子來參與促進(jìn)乳腺瘤形成和轉(zhuǎn)移。 |
|
|
| S7690 |
CK-666
|
CK-666 是肌動(dòng)蛋白相關(guān)蛋白 2/3 (actin-related protein 2/3, Arp2/3) 復(fù)合物的抑制劑,對(duì) BtArp2/3 復(fù)合物和 SpArp2/3 復(fù)合物的 IC50 分別為 17 μM 和 5 μM。 |
- Sci Rep, 2025, 15(1):34331
- Res Sq, 2023, rs.3.rs-3372987
|
|
| F0012 |
β-Actin Antibody [C21N23]
|
ACTB,beta Actin,beta Actin Loading Control,beta-Actin,β-Actin |
- Adv Sci (Weinh), 2025, 12(35):e05725
- Cell Death Dis, 2025, 16(1):672
- J Agric Food Chem, 2025, 73(50):31893-31905
|
|
| F0017 |
α-Smooth Muscle Actin Antibody [L19D14]
|
Actin, alpha-Smooth Muscle,Actin, α-Smooth Muscle,alpha smooth muscle Actin,Alpha-Smooth Muscle Actin,Smooth Muscle Actin,α-Actin,α-Smooth Muscle Actin, α-SMA, a-SMA |
- Bioact Mater, 2024, 34:51-63
- J Plast Surg Hand Surg, 2021, 55(5):284-293
|
|
| F0082 |
Actin Antibody [A24J5]
|
Actin Rabbit mAb recognizes endogenous levels of total Actin protein. |
|
|
| F0440 |
Neurofilament-L Antibody [L10B15]
|
68kDa Neurofilament/NF-L,Neurofilament 68,Neurofilament 70 kDa,Neurofilament-L,NF-L |
|
|
| F0695 |
Neurofilament-M Antibody [H7L9]
|
160 kD Neurofilament Medium,NEFM,Neurofilament 145 kDa,Neurofilament 160,Neurofilament 160 kDa,Neurofilament M,Neurofilament-M |
|
|
| F1648 |
PABP1 Antibody [H6J19]
|
PABP, PABP1 |
|
|
| F0278 |
Cofilin Antibody [D9A5]
|
Cofilin,Cofilin 1 |
|
|
| F2199 |
α Actinin 1/ACTN1 Antibody [C8H2]
|
Actinin alpha,alpha Actinin/ACTN1,alpha-Actinin,α-Actinin |
|
|
| F2226 |
α smooth muscle Actin (acetyl Glu 3) + Actin γ2 (acetyl Glu3) Antibody [H16P9]
|
|
|
|
| F0640 |
N-WASP Antibody [K15N2]
|
N WASP,N-WASP |
|
|
| F0417 |
VASP Antibody [A20G16]
|
|
|
|
| F1962 |
Phospho-Lamin A/C (Ser22) Antibody [D12F9]
|
|
|
|
| F1379 |
Tropomyosin-1 Antibody [G4H1]
|
Tropomyosin (Sarcomeric),Tropomyosin-1 |
|
|
| F2176 |
SUN2 Antibody [D3P18]
|
|
|
|
| F2446 |
γ Actin Antibody [A4H18]
|
gamma Actin,gamma-Actin |
|
|
| F2365 |
Arp3 C-terminal Antibody [F20N23]
|
|
|
|
| F2091 |
Fascin Antibody [N3C10]
|
|
|
|
| F2612 |
ARPC2 Antibody [B10F4]
|
ARPC2,p34-Arc/ARPC2 |
|
|
| F2033 |
α Actinin 4 Antibody [D15C11]
|
alpha Actinin 4,α-Actinin 4 |
|
|
| F2681 |
Cytokeratin 5 Antibody [G20N20]
|
Cytokeratin 5 |
|
|
| F2188 |
Cytokeratin 13 Antibody [L12L19]
|
|
|
|
| F2756 |
CCT2 Antibody [C14D6]
|
|
|
|
| F1440 |
Gelsolin Antibody [D8P23]
|
|
|
|
| F1636 |
Phospho-RAB10 (Thr73) Antibody [M19N14]
|
|
|
|
| F1478 |
Phospho-Zyxin (Ser142/143) Antibody [L24L6]
|
|
|
|
| F2616 |
Cytokeratin 4 Antibody [G16J4]
|
|
|
|