| S0149 |
C-DIM5
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C-DIM5 (DIM-C-pPhOCH3) 是一種孤兒核受體 Nur77 (Nerve growth factor-induced Bα (NGFI-Bα)/nuclear receptor 4A1 (NR4A1)) 的激動(dòng)劑。C-DIM5 (DIM-C-pPhOCH3) 可在RKO結(jié)腸癌細(xì)胞中降低存活率并誘導(dǎo)凋亡。 |
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STAR Protoc, 2025, 6(1):103593
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Cell Rep Med, 2024, S2666-3791(24)00234-9
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Mol Psychiatry, 2022, 10.1038/s41380-022-01497-8
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| S6799 |
DIM-C-pPhOH
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DIM-C-pPhOH (C-DIM8, CDIM8)是一種 nuclear receptor 4A1 (NR4A1)(Nur77) 拮抗劑。DIM-C-pPhOH 可抑制腫瘤生長(zhǎng)和mTOR信號(hào)傳導(dǎo),并誘導(dǎo)細(xì)胞凋亡和細(xì)胞應(yīng)激。DIM-C-pPhOH 可降低細(xì)胞增殖,其對(duì) ACHN細(xì)胞 和 786-O細(xì)胞 的IC50值分別為13.6 μM 和 13.0 μM。 |
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J Adv Res, 2025, S2090-1232(25)00582-X
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Cell Rep, 2024, 43(2):113746
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Mol Psychiatry, 2022, 10.1038/s41380-022-01497-8
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| S6674 |
Cytosporone B (Csn-B)
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Cytosporone B是天然存在的核孤兒受體Nur77(NR4A1) 激動(dòng)劑,EC50為0.278 nM。 |
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Exp Cell Res, 2026, 454(2):114824
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Exp Mol Med, 2025, 57(4):804-819
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J Adv Res, 2025, S2090-1232(25)00582-X
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| F0791New |
Nur77 Antibody [K8J9]
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NGFI-B alpha/Nur77/NR4A1,Nur77 |
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| S6785 |
DIM-C-pPhCO2Me
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DIM-C-pPhCO2Me 是具有抗腫瘤活性的 nuclear receptor 4A1 (NR4A1)(Nur77) 拮抗劑。 |
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