• <dfn id="q240u"></dfn>
      • DYRK1
      • DYRK2
      • DYRK3

      DYRK2 選擇性抑制劑

      目錄號(hào) 產(chǎn)品名 產(chǎn)品描述 Selective / Pan IC50 / Ki
      S3406 LDN-192960 LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively. Selective DYRK2, IC50: 48 nM
      S3817 Harmine hydrochloride Harmine (Telepathine), a fluorescent harmala alkaloid belonging to the beta-carboline family of compounds, is a highly cell-permeant and competitive inhibitor of ATP binding to the kinase pocket of DYRK1A, with about 60-fold higher IC50 value for DYRK2. Harmine also inhibits monoamine oxidases (MAOs), PPARγ and cdc-like kinases (CLKs). Harmine inhibits 5-HT2A serotonin receptor with Ki of 397 nM. Pan DYRK2, IC50: 1.9 μM
      在線咨詢
      聯(lián)系我們
        • <dfn id="q240u"></dfn>
        • 欧美人禽人交片000最新 | 一二三区在线视频 | 女生摸男生的小鸡鸡 | 男人网站 | 亚洲爱爱电影 |