ET-B 拮抗劑
| 目錄號 |
產品名 |
產品描述 |
Selective / Pan |
IC50 / Ki |
| S3051 |
Bosentan Hydrate |
Bosentan (Ro 47-0203) is an endothelin (ET) receptor antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively. |
Pan |
ET-B, Ki: 95 nM |
| S8051 |
Macitentan (ACT 064992) |
Macitentan (ACT 064992) is an orally active, non-peptide, dual ETA/ETB (endothelin) receptor antagonist with IC50 of 0.5 nM/391 nM. |
Pan |
ET-B, IC50: 391 nM |
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