| S1890 |
Nizatidine |
Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM. |
Selective |
Histamine H2 receptor, IC50: 0.9 nM |
| S1880 |
Roxatidine Acetate HCl |
Roxatidine Acetate HCl(HOE 760) is a specific and competitive histamin H2-receptor antagonist, with IC50 of 3.2 μM, inhibits gastric acid secretion and ulcer formation. |
Selective |
Histamine H2 receptor, IC50: 3.2 μM |
| S2065 |
Lafutidine |
Lafutidine (FRG-8813), a newly developed histamine H(2)-receptor antagonist, inhibits gastric acid secretion. |
Selective |
|
| S1845 |
Cimetidine |
Cimetidine (SKF-92334), a histamine congener, competitively inhibits histamine binding to histamine H2 receptors. |
Selective |
|
| S1801 |
Ranitidine Hydrochloride |
Ranitidine (AH19065) is a histamine H2-receptor antagonist, used to treat stomach or intestinal ulcers. |
Selective |
|
| S2078 |
Famotidine |
Famotidine (MK208) is a histamine H2–receptor antagonist with IC50 of 0.6 mM, commonly used to treat heartburn, GERD, ulcers, and other digestive conditions. |
Selective |
|
| S4625 |
Alcaftadine |
Alcaftadine (Lastacaft, R89674) is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines. Alcaftadine is also an antagonist for H2 and H4 receptors with no affinity for the H3 receptor. |
Pan |
H2 receptor, pKi: 7.2 |
| S4117 |
Histamine Phosphate |
Histamine(Histamine diphosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors. |
Pan |
|
| S4118 |
Histamine 2HCl |
Histamine(Ceplene) is an organic nitrogen compound, acts on target cells in mammalian brain via stimulation of Histamine 1/2. |
Pan |
|
