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目錄號(hào)	產(chǎn)品名	產(chǎn)品描述	Selective / Pan	IC50 / Ki
S2480	Loperamide HCl	Loperamide HCl (ADL 2-1294,R-18553 hydrochloride) is a selective μ-opioid receptor agonist opioid with K_i of 3.3 nM, 15-fold and 350-fold selective over the δ subtype and the κ subtype of the opioid receptor, used against diarrhea resulting from gastroenteritis or inflammatory bowel disease.	Selective	μ-opioid receptor, Ki: 3.3 nM
S2103	Naltrexone HCl	Naltrexone HCl(PTI-901) is an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence.	Selective	opioid receptor, IC50: 8 nM
S3066	Naloxone HCl	Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose.	Selective
S2503	Racecadotril	Racecadotril (Acetorphan) is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM.	Selective
S5701	Alvimopan dihydrate (LY246736 dihydrate)	Alvimopan (LY-246736) is a potent, relatively nonselective opioid antagonist with Ki values of 0.77, 4.4, and 40 nM for the μ, δ, and κ opioid receptors, respectively, displaying >100-fold selectivity over other aminergic G-protein-coupled receptors.	Pan	μ-opioid receptor, Ki: 0.77 nM
S5935	Alvimopan	Alvimopan (LY 246736, ADL 8-2698) is a potent, relatively nonselective opioid antagonist with Ki values of 0.77, 4.4, and 40 nM for the μ, δ, and κ opioid receptors, respectively, displaying >100-fold selectivity over other aminergic G-protein-coupled receptors.	Pan	μ-opioid receptor, Ki: 0.77 nM

mumumu-opioid-receptor 選擇性抑制劑 | 激動(dòng)劑 | 拮抗劑