原料藥(僅用于科研)

目錄號(hào)	產(chǎn)品名	產(chǎn)品描述
S3736	Fondaparinux Sodium (Org 31540)	Fondaparinux Sodium (Org 31540, Natural heparin pentasaccharide, Fondaparin, SR-90107A)是一種合成的喃葡萄糖，具有抗血栓形成的活性。它能選擇性地結(jié)合抗凝血酶 III，從而加強(qiáng)對(duì)活化Factor Xa的中和。它是Factor Xa的合成型抑制劑。
S3739	Calcipotriene (MC903)	Calcipotriene (MC903)是calcitriol的合成衍生物，可以誘導(dǎo)角質(zhì)細(xì)胞的分化，抑制其增殖，逆轉(zhuǎn)牛皮癬中角質(zhì)細(xì)胞的異常變化，促使表皮正常生長(zhǎng)。在溶液中不穩(wěn)定，請(qǐng)現(xiàn)配現(xiàn)用！
S3729	Iron sucrose	Iron sucrose (Iron saccharate, Sucroferric oxyhydroxide) is an intravenously administered iron product indicated in the treatment of iron deficiency anemia.
S3730	Metaxalone	Metaxalone (Skelaxin, Methaxalonum, Zorane)是一種肌肉松弛劑，用于放松肌肉、減輕由于拉傷、扭傷和其他原因造成的疼痛。
S3748	Acamprosate Calcium	Acamprosate (N-Acetylhomotaurine, Calcium acetylhomotaurinate,N-acetylhomotaurinate)是一種合成化合物，具有和氨基酸神經(jīng)轉(zhuǎn)運(yùn)體GABA、氨基酸神經(jīng)調(diào)質(zhì)taurine類似的化學(xué)結(jié)構(gòu)。
S1008	Selumetinib (AZD6244)	Selumetinib (AZD6244, ARRY-142886)是一種有效，高選擇性的MEK抑制劑，對(duì)MEK1的IC50為14 nM，對(duì)MEK2的Kd值為530 nM。它也抑制ERK1/2磷酸化，IC50為10 nM，對(duì)p38α， MKK6， EGFR， ErbB2， ERK2， B-Raf等沒(méi)有抑制作用。Selumetinib可抑制細(xì)胞增殖、遷移并誘導(dǎo)凋亡。Phase 3。
S1647	Adenosine	Adenosine是一種核苷，包含腺嘌呤，通過(guò)β-N9-糖苷鍵，與核糖分子（呋喃核糖的）部分連接。
S2475	Imatinib	Imatinib是一種多靶點(diǎn)酪氨酸激酶抑制劑，抑制v-Abl、c-Kit和PDGFR的IC50分別為0.6，0.1和0.1 μM。Imatinib (STI571) 可誘導(dǎo)自噬。
S1833	Butoconazole nitrate	Butoconazole nitrate (RS-35887)是一種抗真菌劑，抑制PHA刺激下人外周血淋巴細(xì)胞中細(xì)胞因子（如IL-2, TNFα, IFN 和 GM-CSF）的分泌，IC50分別為7.2 μg/mL, 14.4 μg/mL, 7.36 μg/mL 和 7.6 μg/mL。
S1282	Artemisinin	Artemisinin青蒿素用于治療耐多藥的惡性瘧疾菌株。
S3207	Iopromide	Iopromide是一種水溶性的親水的非電離的造影劑，用于x-射線成像。
S3727	Vilanterol Trifenate	Vilanterol trifenatate (GW642444M) is a novel inhaled long-acting beta2 adrenoceptor agonist with inherent 24-hour activity for once daily treatment of COPD and asthma.
S3657	Promestriene	Promestriene (3-propyl ethyl, 17B-methyl estradiol) is a synthetic estrogen analog that has been reported to significantly improve the symptoms of vaginal atrophy caused by estrogen deprivation in topical application.
S3673	Sulfaphenazole	Sulfaphenazole (Depocid, Depotsulfonamide, Plisulfan, Raziosulfa) is an inhibitor of CYP2C9 with Ki value of 0.3 μM and demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki values of 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19).
S3726	Selexipag	Selexipag (NS-304, ACT-293987) is an orally active, first-in-class, selective prostacyclin IP receptor agonist with Ki value of 260 nM for human IP, whereas Ki values > 10,000 nM are measured at the other human G-protein-coupled prostanoid receptors (EP1-4, DP, FP and TP).
S3728	Grazoprevir	Grazoprevir anhydrous (MK5172) 是一種 Hepatitis C Virus NS3/4A Protease 的抑制劑，HCV genotype 1a、1B和4的IC50值分別為7pM、4pM和62pM。
S3731	Tipiracil hydrochloride	Tipiracil (MA-1)是一種 thymidine phosphorylase的抑制劑，該酶可將三氟吡啶降解為三氟胸苷。它與三氟吡啶的組合可增加三氟吡啶的生物利用度。
S3671	Quinestrol	Quinestrol (Ethinylestradiol 3-cyclopentyl ether, EE2CPE, W-3566) is a synthetic, steroidal estrogen which is used in hormone replacement therapy and occasionally to treat breast cancer and prostate cancer.
S3667	Imipenem	Imipenem acts as an inhibitor of AmpC β-lactamase and is an antibiotic useful for the treatment of a number of bacterial infections.
S3716	Flibanserin	Flibanserin (BIMT-17, BIMT-17-BS) 是一種非激素類、作用于中樞的小分子，是突觸后5-HT1A受體的激動(dòng)劑，也是5-HT2A的拮抗劑。

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