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    • 原料藥(僅用于科研)

      目錄號 產(chǎn)品名 產(chǎn)品描述
      S4833 Cefoxitin sodium Cefoxitin Sodium is the sodium salt form of cefoxitin, a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.
      S1491 Fludarabine Fludarabine在血管平滑肌細(xì)胞中是一種STAT1活化抑制劑,特異性降低STAT1蛋白質(zhì)水平(和mRNA水平) ,而對其他STATs無此作用。它還是一種DNA合成抑制劑。Fludarabine可誘導(dǎo)凋亡。
      S5563 Thioridazine hydrochloride Thioridazine (Aldazine, Mellaril) is a potent antianxiety and antipsychotic agent.
      S5430 Metoprolol Metoprolol is a cardioselective β1-adrenergic blocking agent with log Kd values of ?7.26±0.07, ?6.89±0.09, ?5.16±0.12 for β1, β2, and β3 adrenoceptors, respectively. It is used for acute myocardial infarction, heart failure, angina pectoris and mild to moderate hypertension.
      S5517 Fenamic acid Fenamic acid (N-Phenylanthranilic acid, 2-(Phenylamino)benzoic acid, 2-Anilinobenzoic acid, Diphenylamine-2-carboxylic acid) serves as a parent structure for several nonsteroidal anti-inflammatory drugs (NSAIDs), including mefenamic acid, tolfenamic acid, flufenamic acid, and meclofenamic acid.
      S5433 Sodium succinate Sodium succinate (Sodium 3-carboxypropanoate, Disodium butanedioate) is the sodium salt form of succinate, which is an important metabolite at the cross-road of several metabolic pathways and involved in the formation and elimination of reactive oxygen species.
      S4129 Sevelamer HCl Sevelamer是一種磷酸鹽結(jié)合的藥物,用于治療慢性腎臟疾病的高磷酸鹽血癥。
      S1393 Pirarubicin Pirarubicin是一種蒽環(huán)類抗生素,同時(shí)也是一種DNA/RNA合成抑制劑,摻入DNA并與topoisomerase II相互作用,是一種抗腫瘤藥物。
      S1614 Riluzole Riluzole是谷氨酸鹽釋放抑制劑,具有神經(jīng)保護(hù)、抗癲癇、抗焦慮以及麻醉作用。
      S3041 Droxidopa Droxidopa (L-DOPS)是一種精神藥物,是合成的氨基酸前體,它作為神經(jīng)傳導(dǎo)物質(zhì)去甲腎上腺素和腎上腺素的前藥來發(fā)揮作用。
      S5281 Dapiprazole Hydrochloride Dapiprazole Hydrochloride (Glamidolo Hydrochloride, Reversil Hydrochloride) is the hydrochloride salt form of dapiprazole, an alpha-adrenergic blocker used to reverse mydriasis after eye examination.
      S5297 Vidarabine monohydrate Vidarabine (Spongoadenosine, Vira-A) is a nucleoside antibiotic with antiviral acitivity that interferes with the synthesis of viral DNA. It is used to treat herpes simplex and varicella zoster viruses.
      S3081 Ulipristal Acetate (CDB 2914) Ulipristal acetate (CDB-2914, HRP 2000, RU 44675)是一種選擇性的孕酮受體調(diào)節(jié)劑(SPRM),用于無保護(hù)措施性交或避孕失敗后120小時(shí)(5 天)內(nèi)的緊急避孕。
      S2597 Oseltamivir Phosphate Oseltamivir Phosphate(Tamiflu) 是一種有效的和選擇性的,甲型流感和乙型流感病毒復(fù)制必需的神經(jīng)氨酸酶的抑制劑,用于治療流行性感冒。
      S5243 Ruxolitinib (INCB18424) Phosphate Ruxolitinib Phosphate (INCB018424, INC424)是Ruxolitinib的磷酸鹽形式。Ruxolitinib 是第一個(gè)應(yīng)用于臨床的,有效的,選擇性JAK1/2抑制劑,在無細(xì)胞試驗(yàn)中IC50為3.3 nM/2.8 nM。作用于JAK1,JAK2與作用于JAK3相比,選擇性高130多倍。Ruxolitinib 通過毒性線粒體自噬殺死腫瘤細(xì)胞。Ruxolitinib 可誘導(dǎo)自噬并增強(qiáng)細(xì)胞凋亡。
      S5402 Dasabuvir (ABT-333) Dasabuvir (ABT-333) is a non-nucleoside inhibitor of NS5B viral RNA-dependent RNA polymerase that inhibits recombinant NS5B polymerases derived from HCV genotype 1a and 1b clinical isolates with IC50 values between 2.2 and 10.7 nM. It is at least 7,000-fold selective for the inhibition of HCV genotype 1 polymerases over human/mammalian polymerases.
      S5257 Doxapram Doxapram is a central respiratory stimulant with a brief duration of action.
      S1398 Stavudine (d4T) Stavudine (d4T, BMY-27857, Sanilvudine, NSC 163661)是一種核苷類似物逆轉(zhuǎn)錄酶抑制劑(NARTI),有效作用于HIV。
      S4082 Spiramycin Spiramycin (Formacidine) 是16元環(huán)大環(huán)內(nèi)酯(抗生素)。
      S1379 Isotretinoin (13-cis retinoic acid) Isotretinoin (13-cis retinoic acid)被開發(fā)用作治療腦癌、胰腺癌等的化療藥物。
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