| S4833 |
Cefoxitin sodium |
Cefoxitin Sodium is the sodium salt form of cefoxitin, a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity. |
| S1491 |
Fludarabine |
Fludarabine在血管平滑肌細(xì)胞中是一種STAT1活化抑制劑,特異性降低STAT1蛋白質(zhì)水平(和mRNA水平) ,而對其他STATs無此作用。它還是一種DNA合成抑制劑。Fludarabine可誘導(dǎo)凋亡。 |
| S5563 |
Thioridazine hydrochloride |
Thioridazine (Aldazine, Mellaril) is a potent antianxiety and antipsychotic agent. |
| S5430 |
Metoprolol |
Metoprolol is a cardioselective β1-adrenergic blocking agent with log Kd values of ?7.26±0.07, ?6.89±0.09, ?5.16±0.12 for β1, β2, and β3 adrenoceptors, respectively. It is used for acute myocardial infarction, heart failure, angina pectoris and mild to moderate hypertension. |
| S5517 |
Fenamic acid |
Fenamic acid (N-Phenylanthranilic acid, 2-(Phenylamino)benzoic acid, 2-Anilinobenzoic acid, Diphenylamine-2-carboxylic acid) serves as a parent structure for several nonsteroidal anti-inflammatory drugs (NSAIDs), including mefenamic acid, tolfenamic acid, flufenamic acid, and meclofenamic acid. |
| S5433 |
Sodium succinate |
Sodium succinate (Sodium 3-carboxypropanoate, Disodium butanedioate) is the sodium salt form of succinate, which is an important metabolite at the cross-road of several metabolic pathways and involved in the formation and elimination of reactive oxygen species. |
| S4129 |
Sevelamer HCl |
Sevelamer是一種磷酸鹽結(jié)合的藥物,用于治療慢性腎臟疾病的高磷酸鹽血癥。 |
| S1393 |
Pirarubicin |
Pirarubicin是一種蒽環(huán)類抗生素,同時(shí)也是一種DNA/RNA合成抑制劑,摻入DNA并與topoisomerase II相互作用,是一種抗腫瘤藥物。 |
| S1614 |
Riluzole |
Riluzole是谷氨酸鹽釋放抑制劑,具有神經(jīng)保護(hù)、抗癲癇、抗焦慮以及麻醉作用。 |
| S3041 |
Droxidopa |
Droxidopa (L-DOPS)是一種精神藥物,是合成的氨基酸前體,它作為神經(jīng)傳導(dǎo)物質(zhì)去甲腎上腺素和腎上腺素的前藥來發(fā)揮作用。 |
| S5281 |
Dapiprazole Hydrochloride |
Dapiprazole Hydrochloride (Glamidolo Hydrochloride, Reversil Hydrochloride) is the hydrochloride salt form of dapiprazole, an alpha-adrenergic blocker used to reverse mydriasis after eye examination. |
| S5297 |
Vidarabine monohydrate |
Vidarabine (Spongoadenosine, Vira-A) is a nucleoside antibiotic with antiviral acitivity that interferes with the synthesis of viral DNA. It is used to treat herpes simplex and varicella zoster viruses. |
| S3081 |
Ulipristal Acetate (CDB 2914) |
Ulipristal acetate (CDB-2914, HRP 2000, RU 44675)是一種選擇性的孕酮受體調(diào)節(jié)劑(SPRM),用于無保護(hù)措施性交或避孕失敗后120小時(shí)(5 天)內(nèi)的緊急避孕。 |
| S2597 |
Oseltamivir Phosphate |
Oseltamivir Phosphate(Tamiflu) 是一種有效的和選擇性的,甲型流感和乙型流感病毒復(fù)制必需的神經(jīng)氨酸酶的抑制劑,用于治療流行性感冒。 |
| S5243 |
Ruxolitinib (INCB18424) Phosphate |
Ruxolitinib Phosphate (INCB018424, INC424)是Ruxolitinib的磷酸鹽形式。Ruxolitinib 是第一個(gè)應(yīng)用于臨床的,有效的,選擇性JAK1/2抑制劑,在無細(xì)胞試驗(yàn)中IC50為3.3 nM/2.8 nM。作用于JAK1,JAK2與作用于JAK3相比,選擇性高130多倍。Ruxolitinib 通過毒性線粒體自噬殺死腫瘤細(xì)胞。Ruxolitinib 可誘導(dǎo)自噬并增強(qiáng)細(xì)胞凋亡。 |
| S5402 |
Dasabuvir (ABT-333) |
Dasabuvir (ABT-333) is a non-nucleoside inhibitor of NS5B viral RNA-dependent RNA polymerase that inhibits recombinant NS5B polymerases derived from HCV genotype 1a and 1b clinical isolates with IC50 values between 2.2 and 10.7 nM. It is at least 7,000-fold selective for the inhibition of HCV genotype 1 polymerases over human/mammalian polymerases. |
| S5257 |
Doxapram |
Doxapram is a central respiratory stimulant with a brief duration of action. |
| S1398 |
Stavudine (d4T) |
Stavudine (d4T, BMY-27857, Sanilvudine, NSC 163661)是一種核苷類似物逆轉(zhuǎn)錄酶抑制劑(NARTI),有效作用于HIV。 |
| S4082 |
Spiramycin |
Spiramycin (Formacidine) 是16元環(huán)大環(huán)內(nèi)酯(抗生素)。 |
| S1379 |
Isotretinoin (13-cis retinoic acid) |
Isotretinoin (13-cis retinoic acid)被開發(fā)用作治療腦癌、胰腺癌等的化療藥物。 |