原料藥(僅用于科研)

目錄號	產(chǎn)品名	產(chǎn)品描述
S3046	Azilsartan	Azilsartan (TAK-536)是angiotensin II type 1 (AT1)（血管緊張素II 1型）受體拮抗劑，IC50為2.6 nM。
S5353	Cefpiramide sodium	Cefpiramide sodium (CPMS, SM-1652,wy-44635) is an anionic β-lactam antibiotic. It exhibits antibacterial activity against gram-positive and gram-negative bacteria, in particular, to Pseudomonas aeruginosa, which can result in achronic life-threatening infection in the lungs of cystic fibrosis patients.
S5651	Dexrazoxane	Dexrazoxane (ICRF-187) is an anticancer drug able to block mitosis and to arrest dividing cells. It is an iron chelator and provides cardioprotection against anthracycline toxicity.
S5647	Emedastine Difumarate	Emedastine Difumarate (Rapimine, Emedastine fumarate) is the difumarate salt form of emedastine, a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
S5253	Cisapride (R 51619)	Cisapride (R 51619, Kaudalit, Kinestase, Prepulsid, Presid, Pridesia, Propulsid) is a nonselective 5-HT4 receptor agonist with gastroprokinetic effects.
S5500	Amodiaquine hydrochloride	Amodiaquine Hydrochloride is the hydrochloride salt of amodiaquine, an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory properties.
S5537	Tizanidine	Tizanidine is an imidazoline derivative and a centrally acting α2 adrenergic agonist used as a muscle relaxant for therapy of acute muscle spasms and chronic spasticity.
S5621	Cilastatin	Cilastatin(MK0791) is a renal dehydropeptidase-I and leukotriene D4 dipeptidase inhibitor.
S1655	Ezetimibe (SCH-58235)	Ezetimibe (SCH-58235) 是一種有效的、選擇性的膽固醇吸收抑制劑，用來降低膽固醇。
S5540	Landiolol hydrochloride	Landiolol hydrochloride (ONO-1101) is the hydrochloride salt form of Landiolol, which is an ultra-short-acting β1 selective adrenoceptor antagonist.
S5624	Paliperidone Palmitate	Paliperidone Palmitate (9-hydroxyrisperidone palmitate) is a palmitate ester of paliperidone, which is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class.
S5623	Bedaquiline	Bedaquiline (TMC-207, R207910), a diarylquinoline, binds to subunit c of mycobacterial ATP synthase and inhibits its activity. It is highly selective for mycobacterial ATP synthase enzyme compared to homologous eukaryotic enzyme (Selectivity Index >20 000).
S5413	Ertugliflozin	Ertugliflozin (MK-8835, PF-04971729) is a potent and selective sodium-dependent glucose cotransporter 2 inhibitor with IC50 values of 0.877 nM for h-SGLT2 and 1000-fold higher for h-SGLT1.
S5482	Prilocaine hydrochloride	Prilocaine hydrochloride is the hydrochloride salt form of prilocaine, which is a local anesthetic.
S5358	Regadenoson	Regadenoson (CVT-3146, Lexiscan) is a selective A2A adenosine receptor agonist with coronary vasodilating activity.
S5357	Safinamide	Safinamide (EMD-1195686, PNU-15774E) is an orally active, selective, reversible monoamine oxidase-B inhibitor with both dopaminergic and non-dopaminergic (glutamatergic) properties. The IC50 value of safinamide for MAO-B is 98 nM.
S5240	Lenvatinib Mesylate	Lenvatinib Mesylate是一種合成、具有口服活性的 tyrosine kinase 的抑制劑，可抑制血管內(nèi)皮生長因子受體(VEGFR1-3)，成纖維細胞生長因子受體(FGFR1-4)，血小板衍生生長因子受體(PDGFRα)，干細胞因子受體(Kit (c-Kit))，并在轉(zhuǎn)染過程中重新排列(RET (c-RET))。甲磺酸來伐替尼具有潛在的抗腫瘤活性。
S5239	Paroxetine mesylate	Paroxetine Mesylate(BRL-29060A mesylate,FG-7051 mesylate) is the mesylate salt form of paroxetine, a phenylpiperidine derivative and a selective serotonin reuptake inhibitor (SSRI) with antidepressant and anxiolytic properties.
S5205	Nilotinib hydrochloride	Nilotinib hydrochloride (AMN-107) is the hydrochloride salt form of nilotinib, an orally bioavailable Bcr-Abl tyrosine kinase inhibitor with antineoplastic activity.
S2868	Alogliptin (SYR-322) benzoate	Alogliptin (SYR-322) benzoate是一種有效的，選擇性的DPP-4抑制劑，IC50為<10 nM，比作用于DPP-8和DPP-9選擇性高10000倍以上。

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